Q9Y468 | LMBL1_HUMAN | Lethal(3)malignant brain tumor-like protein 1 (L3MBTL1)

Pfam Domain Table

AccessionDomainRangeColor
PF01530zf-C2HC - Zinc finger, C2HC type621~649
PF02820MBT - mbt repeat310~378
PF02820MBT - mbt repeat417~484
PF02820MBT - mbt repeat521~587

3D structures mapped by conservation among orthologs

[ Domain: "SH3" // MBT ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL3351077 IC50 = 98.0 nM 532.56 NC(=O)c1cc[n+](CC2=C(C(=O)[O-])N3C(=O)[C@@H](NC(=O)[C@@H](c4ccccc4)S(=O)(=O)O)[C@H]3SC2)cc1 Homo sapiens CHEMBL4138803 single protein format
CHEMBL1257003 IC50 = 282.0 nM 437.19 COc1cc(/C=C(\C#N)C(=O)c2ccc(O)c(O)c2)cc(I)c1O Homo sapiens CHEMBL4138803 single protein format
CHEMBL2426365 IC50 = 740.0 nM 543.76 O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c(NCc2ccccc2)c1)N1CCC(N2CCCC2)CC1 Homo sapiens CHEMBL2429078 single protein format