Q9UPE1 | SRPK3_HUMAN | SRSF protein kinase 3 (SRPK3)

Helixβ‑strandTurn secondary structure

Pfam Domain Table

AccessionDomainRangeColor
PF00069Pkinase79–221
PF00069Pkinase388–565

 3D structures mapped by conservation among orthologs


 [ Alpha Fold Model ] (go)



 Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL4468747 IC50 = 4.81 nM 472.54 CCc1cc2c(cc1-c1cccc(S(=O)(=O)F)c1)C(C)(C)c1[nH]c3cc(C#N)ccc3c1C2=O Homo sapiens CHEMBL5321381 single protein format
CHEMBL4064277 IC50 = 27.0 nM 349.36 O=C(Nc1cc(C(F)(F)F)ccc1N1CCCCC1)c1ccncc1 Homo sapiens CHEMBL5321381 single protein format
CHEMBL5085558 IC50 = 40.0 nM 461.91 CN(c1ncccc1CNc1ccnc(-c2nc3c(F)c(Cl)ccc3[nH]2)n1)S(C)(=O)=O Homo sapiens CHEMBL5058560 single protein format
CHEMBL5074274 IC50 = 166.0 nM 507.52 O=C(Nc1cc(C(F)(F)F)ccc1N1CCN(Cc2ccccn2)CC1)c1ccc(-c2ccncc2)o1 Homo sapiens CHEMBL5321381 single protein format