Q9UIF8 | BAZ2B_HUMAN | Bromodomain adjacent to zinc finger domain protein 2B (BAZ2B)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00439 | Bromodomain - Bromodomain | 2069~2148 | |
PF00628 | PHD - PHD-finger | 1934~1978 | |
PF01429 | MBD - Methyl-CpG binding domain | 740~812 | |
PF02791 | DDT - DDT domain | 1089~1149 | |
PF15613 | WSD - Williams-Beuren syndrome DDT (WSD), D-TOX E motif | 1373~1403 |
3D structures mapped by conservation among orthologs
[ Domain: "Bromodomain" // Bromodomain ]
- 2E7O
- 3G0L
- 3Q2F
- 4CUP
- 4CUQ
- 4CUR
- 4CUS
- 4CUT
- 4CUU
- 4IR3
- 4IR4
- 4IR5
- 4IR6
- 4NR9
- 4NRA
- 4NRB
- 4NRC
- 4QC1
- 4QC3
- 4RVR
- 4XUA
- 4XUB
- 5CQ3
- 5CQ4
- 5CQ5
- 5CQ6
- 5CQ7
- 5CQ8
- 5CQA
- 5CU8
- 5CUA
- 5CUB
- 5CUC
- 5CUD
- 5CUE
- 5CUG
- 5DYU
- 5DYX
- 5E73
- 5E74
- 5E9I
- 5E9K
- 5E9L
- 5E9M
- 5E9Y
- 5L8T
- 5L8U
- 5L96
- 5L97
- 5L98
- 5L99
- 5MGE
- 5MGF
- 5MGG
- 5OR9
- 5ORB
- 5PB7
- 5PB8
- 5PB9
- 5PBA
- 5PBB
- 5PBC
- 5PBD
- 5PBE
- 5PBF
- 5PBG
- 5PBH
- 5PBI
- 5PBJ
- 5PBK
- 5PBL
- 5PBM
- 5PBN
- 5PBO
- 5PBP
- 5PBQ
- 5PBR
- 5PBS
- 5PBT
- 5PBU
- 5PBV
- 5PBW
- 5PBX
- 5PBY
- 5PBZ
- 5PC0
- 5PC1
- 5PC2
- 5PC3
- 5PC4
- 5PC5
- 5PC6
- 5PC7
- 5PC8
- 5PC9
- 5PCA
- 5PCB
- 5PCC
- 5PCD
- 5PCE
- 5PCF
- 5PCG
- 5PCH
- 5PCI
- 5PCJ
- 5PCK
- 5PCL
- 5PCM
- 5PCN
- 5PCO
- 5PCP
- 5PCQ
- 5PCR
- 5PCS
- 5PCT
- 5PCU
- 5PCV
- 5PCW
- 5PCX
- 5PCZ
- 5PD0
- 5PD1
- 5PD2
- 5PD3
- 5PD4
- 5PD5
- 5PD6
- 5PD7
- 5PD8
- 5PD9
- 5PDA
- 5PDB
- 5PDC
- 5PDD
- 5PDE
- 5PDF
- 5PDG
- 5PDH
- 5PDI
- 5PDJ
- 5PDK
- 5PDL
- 5PDM
- 5PDN
- 5PDO
- 5PDP
- 5PDQ
- 5PDR
- 5PDS
- 5PDT
- 5PDU
- 5PDV
- 5PDW
- 5PDX
- 5PDY
- 5PDZ
- 5PE0
- 5PE1
- 5PE2
- 5PE3
- 5PE4
- 5PE5
- 5PE6
- 5PE7
- 5PE8
- 5PE9
- 5PEA
- 5PEB
- 5PEC
- 5PED
- 5PEE
- 5PEF
- 5PEG
- 5PEH
- 5PEI
- 5PEJ
- 5PEK
- 5PEL
- 5PEM
- 5PEN
- 5PEO
- 5PEQ
- 5PER
- 5PES
- 5PET
- 5PEU
- 5PEV
- 5PEW
- 5PEX
- 5PEY
- 5PEZ
- 5PF0
- 5PF1
- 5PF2
- 5PF3
- 5PF4
- 5PF5
- 5PF6
- 5PF7
- 5PF8
- 5PF9
- 5PFA
- 5PFB
- 5PFC
- 5PFD
- 5PFE
- 5PFF
- 5PFG
- 5PFH
- 5PFI
- 5PFJ
- 5PFL
- 5PFM
- 5PFN
- 5PFO
- 5PFP
- 5PFQ
- 5PFR
- 5PFS
- 5PFT
- 5PFU
- 5PFV
- 5PFW
- 5PFX
- 5PFY
- 5PFZ
- 5PG0
- 5PG1
- 5PG2
- 5PG3
- 5PG4
- 5PG5
- 5PG6
- 5PG7
- 5PG8
- 5PG9
- 5PGA
- 5PGB
- 5PGC
- 5PGD
- 5PGE
- 5PGF
- 5PGG
- 5PGH
- 5PGI
- 5PGJ
- 5PGK
- 5PGL
- 5PGN
- 5PGO
- 5PGP
- 5PGQ
- 5PGR
- 5PGS
- 5PGT
- 6FGT
- 6FGU
- 6FH6
- 6FH7
[ Domain: "FYVE/PHD zinc finger" // PHD_1 ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL4296718 | IC50 | = | 180.0 | nM | 357.42 | Cn1cc(CCn2cnc(-c3cnn(C)c3)c2-c2ccc(C#N)cc2)cn1 | Homo sapiens | CHEMBL3419225 | single protein format | |
CHEMBL3771216 | IC50 | = | 370.0 | nM | 279.34 | CC(=O)c1cc(-c2ccccc2CO)c2cc(C)ccn12 | Homo sapiens | CHEMBL3772736 | assay format | |
CHEMBL3770155 | IC50 | = | 410.0 | nM | 295.34 | COc1ccn2c(C(C)=O)cc(-c3ccccc3CO)c2c1 | Homo sapiens | CHEMBL3772736 | assay format | |
CHEMBL3739699 | IC50 | = | 430.0 | nM | 371.46 | CCCOc1ccn2c(C(C)=O)cc(-c3ccccc3S(C)(=O)=O)c2c1 | Homo sapiens | CHEMBL3772736 | assay format | |
CHEMBL3770449 | IC50 | = | 540.0 | nM | 350.42 | CC(=O)c1cc(-c2ccccc2CO)c2cc(N3CCOCC3)ccn12 | Homo sapiens | CHEMBL3772736 | assay format | |
CHEMBL3770493 | IC50 | = | 610.0 | nM | 357.41 | CC(=O)c1cc(-c2ccccc2CO)c2cc(Oc3ccccc3)ccn12 | Homo sapiens | CHEMBL3772736 | assay format | |
CHEMBL3770199 | IC50 | = | 670.0 | nM | 442.54 | CC(=O)c1cc(-c2ccccc2S(C)(=O)=O)c2cc(CNC(=O)OC(C)(C)C)ccn12 | Homo sapiens | CHEMBL3772736 | assay format | |
CHEMBL3415184 | IC50 | = | 770.0 | nM | 362.37 | Cc1cn(Cn2cnc(-c3cnn(C)c3)c2-c2ccc(C#N)cc2F)nn1 | Homo sapiens | CHEMBL3419225 | single protein format | |
CHEMBL3415185 | IC50 | = | 790.0 | nM | 362.37 | Cc1cn(Cn2cnc(-c3cnn(C)c3)c2-c2ccc(C#N)c(F)c2)nn1 | Homo sapiens | CHEMBL3419225 | single protein format | |
CHEMBL3770214 | IC50 | = | 820.0 | nM | 343.4 | COc1ccn2c(C(C)=O)cc(-c3ccccc3S(C)(=O)=O)c2c1 | Homo sapiens | CHEMBL3772736 | assay format | |
CHEMBL3770277 | IC50 | = | 840.0 | nM | 405.48 | CC(=O)c1cc(-c2ccccc2S(C)(=O)=O)c2cc(Oc3ccccc3)ccn12 | Homo sapiens | CHEMBL3772736 | assay format | |
CHEMBL3770112 | IC50 | = | 1000.0 | nM | 265.31 | CC(=O)c1cc(-c2ccccc2CO)c2ccccn12 | Homo sapiens | CHEMBL3772736 | assay format | |
CHEMBL4069412 | Ki | = | 840.0 | nM | 377.29 | CN1C[C@H](Nc2cnn(C)c(=O)c2Br)C[C@H](c2ccccc2)C1 | Homo sapiens | CHEMBL5214219 | single protein format |