Q9P0G3 | KLK14_HUMAN | Kallikrein-14 (KLK14)

Pfam Domain Table

AccessionDomainRangeColor
PF00089Trypsin - Trypsin41~260

3D structures mapped by conservation among orthologs


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL4206734 IC50 = 8.0 nM 458.52 Cc1nn(-c2ccccc2)c(C)c1NC(=O)COC(=O)Cc1c(C)[nH]c2cc(C(=N)N)ccc12 Homo sapiens CHEMBL4201847 assay format
CHEMBL4575974 IC50 = 100.0 nM 327.34 CCOc1cc2c(=O)oc(-c3ccccc3OC)nc2cc1OC Homo sapiens CHEMBL4424187 single protein format
CHEMBL1580091 IC50 = 970.0 nM 329.81 CSc1nc(-c2ccc(Cl)cc2)nn1C(=O)c1ccccc1 Homo sapiens CHEMBL2412648 single protein format