Q9NSD7 | RL3R1_HUMAN | Relaxin-3 receptor 1 (RXFP3)
Helixβ‑strandTurn secondary structure
Pfam Domain Table
| Accession | Domain | Range | Color |
|---|---|---|---|
| PF00001 | 7tm_1 | 98–196 | |
| PF00001 | 7tm_1 | 214–389 |
3D structures mapped by conservation among orthologs
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
| molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
|---|---|---|---|---|---|---|---|---|---|---|
| CHEMBL5089949 |  |
Ki | = | 68.7 | nM | 402.46 | COC(=O)c1ccc(CCNC(=N)N/N=C/c2c[nH]c3c(C)cc(C#N)cc23)cc1 | Homo sapiens | CHEMBL5033954 | cell-based format |
| CHEMBL5094670 |  |
Ki | = | 268.0 | nM | 374.45 | COc1cc(C)c2[nH]cc(/C=N/NC(=N)NCCc3ccc(C#N)cc3)c2c1 | Homo sapiens | CHEMBL5033954 | cell-based format |
| CHEMBL4522365 |  |
Ki | = | 274.0 | nM | 383.88 | CCc1cc(O)cc2c(/C=N/NC(=N)NCCc3ccc(Cl)cc3)c[nH]c12 | Homo sapiens | CHEMBL5033954 | cell-based format |