Q9HCP0 | KC1G1_HUMAN | Casein kinase I isoform gamma-1 (CSNK1G1)
Pfam Domain Table
| Accession | Domain | Range | Color |
|---|---|---|---|
| PF00069 | Pkinase - Protein kinase domain | 45~262 | |
| PF12605 | CK1gamma_C - Casein kinase 1 gamma C terminal | 331~362 | |
| PF12605 | CK1gamma_C - Casein kinase 1 gamma C terminal | 369~392 |
3D structures mapped by conservation among orthologs
[ Domain: "Protein kinase" // Pkinase_Tyr ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
| molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
|---|---|---|---|---|---|---|---|---|---|---|
| CHEMBL511410 |  |
IC50 | = | 160.0 | nM | 338.32 | NC(=O)C(Nc1c(Nc2ccncc2)c(=O)c1=O)c1cccc(O)c1 | Homo sapiens | CHEMBL1011428 | single protein format |
| CHEMBL466496 |  |
IC50 | = | 250.0 | nM | 293.33 | C[C@@H](Nc1c(Nc2ccncc2)c(=O)c1=O)c1ccccc1 | Homo sapiens | CHEMBL1011428 | single protein format |
| CHEMBL4744428 |  |
IC50 | <= | 500.0 | nM | 433.52 | CC(C)n1cnnc1-c1cccc(NC(=O)[C@H]2CN(c3ccc(C4CC4)nc3)CCO2)n1 | Homo sapiens | CHEMBL4727567 | single protein format |
| CHEMBL467079 |  |
IC50 | = | 520.0 | nM | 322.32 | NC(=O)C(Nc1c(Nc2ccncc2)c(=O)c1=O)c1ccccc1 | Homo sapiens | CHEMBL1011428 | single protein format |