Q9H792 | PEAK1_HUMAN | Inactive tyrosine-protein kinase PEAK1 (PEAK1)
Pfam Domain Table
| Accession | Domain | Range | Color |
|---|---|---|---|
| PF00069 | Pkinase - Protein kinase domain | 1477~1659 |
3D structures mapped by conservation among orthologs
[ Domain: "split helical dimerization (SHED) domain" // UNK_F_TYPE ]
[ Domain: "Protein kinase" // Pkinase_Tyr ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
| molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
|---|---|---|---|---|---|---|---|---|---|---|
| CHEMBL388978 |  |
IC50 | = | 3.04 | nM | 466.54 | CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 | Homo sapiens | CHEMBL4328552 | single protein format |
| CHEMBL5279425 |  |
IC50 | = | 620.0 | nM | 381.46 | O=C(c1ccc2c(c1)OCCO2)C1CCN(c2ncnc3sccc23)CC1 | Homo sapiens | CHEMBL5248033 | single protein format |