Q9GZN0 | GPR88_HUMAN | Probable G-protein coupled receptor 88 (GPR88)
Helixβ‑strandTurn secondary structure
Pfam Domain Table
| Accession | Domain | Range | Color |
|---|---|---|---|
| PF00001 | 7tm_1 | 49–336 |
3D structures mapped by conservation among orthologs
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
| molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
|---|---|---|---|---|---|---|---|---|---|---|
| CHEMBL3403780 |  |
Ki | = | 219.0 | nM | 368.52 | CCCC(C)COc1ccc([C@H](CN)NC(=O)[C@@H](C)c2ccccc2)cc1 | Homo sapiens | CHEMBL5240736 | single protein format |
| CHEMBL4595209 |  |
Ki | = | 224.0 | nM | 459.59 | COCc1ccc(-c2ccc(N(C[C@@H](N)[C@@H](C)OC)C(=O)[C@@H]3C[C@H]3c3ccccn3)cc2)cc1 | Homo sapiens | CHEMBL5240736 | single protein format |
| CHEMBL3401461 |  |
Ki | = | 277.0 | nM | 455.65 | CCCc1ccc(-c2ccc(N(C[C@@H](N)[C@@H](C)CC)C(=O)[C@@H]3C[C@H]3c3ccccn3)cc2)cc1 | Homo sapiens | CHEMBL5240736 | single protein format |
| CHEMBL5285428 |  |
Ki | = | 487.0 | nM | 455.65 | CCCc1ccc(-c2ccc(N(C[C@@H](N)[C@@H](C)CC)C(=O)[C@H]3C[C@@H]3c3ccccn3)cc2)cc1 | Homo sapiens | CHEMBL5240736 | single protein format |
| CHEMBL3403768 |  |
Ki | = | 612.0 | nM | 369.51 | CCCC(C)COc1ccc([C@H](CO)NC(=O)[C@@H](C)c2ccccc2)cc1 | Homo sapiens | CHEMBL5240736 | single protein format |