Q99759 | M3K3_HUMAN | Mitogen-activated protein kinase kinase kinase 3 (MAP3K3)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00069 | Pkinase - Protein kinase domain | 364~621 | |
PF00564 | PB1 - PB1 domain | 45~120 |
3D structures mapped by conservation among orthologs
[ Domain: "Ubiquitin-like" // PB1 ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL388978 | IC50 | = | 10.9 | nM | 466.54 | CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 | Homo sapiens | CHEMBL4328493 | single protein format | |
CHEMBL4554938 | IC50 | = | 34.8 | nM | 416.49 | CN1C(=O)c2sccc2N(C)c2nc(Nc3ccc(S(N)(=O)=O)cc3)ncc21 | Homo sapiens | CHEMBL5212984 | single protein format |