Q99594 | TEAD3_HUMAN | Transcriptional enhancer factor TEF-5 (TEAD3)
Helixβ‑strandTurn secondary structure
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF01285 | TEA | 32–98 | |
PF17725 | YBD | 223–432 |
3D structures mapped by conservation among orthologs
[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // KOG3841 ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL5422959 | IC50 | = | 3.0 | nM | 406.39 | C=CC(=O)N1CC(c2nc(-c3ccc(OC(F)(F)F)cc3)c3ncsc3n2)C1 | Homo sapiens | CHEMBL5369244 | single protein format | |
CHEMBL5401444 | IC50 | = | 4.0 | nM | 403.36 | C=CC(=O)N1CC(c2nc(-c3ccc(OC(F)(F)F)cc3)c3ncn(C)c3n2)C1 | Homo sapiens | CHEMBL5369244 | single protein format | |
CHEMBL5408536 | IC50 | = | 4.0 | nM | 426.78 | C=C(Cl)C(=O)NCc1nn(-c2ccc(OC(F)(F)F)cc2)c2nccc(CO)c12 | Homo sapiens | CHEMBL5374058 | single protein format | |
CHEMBL5438256 | IC50 | = | 4.0 | nM | 397.78 | CN(Cc1nn(-c2ccc(OC(F)(F)F)cc2)c2ccccc12)C(=O)CCl | Homo sapiens | CHEMBL5374058 | single protein format | |
CHEMBL5411200 | IC50 | = | 5.0 | nM | 412.37 | C#Cc1ccnc2c1c(C1CN(C(=O)C=C)C1)nn2-c1ccc(OC(F)(F)F)cc1 | Homo sapiens | CHEMBL5374058 | single protein format | |
CHEMBL5415215 | IC50 | = | 7.0 | nM | 407.39 | C=CC(=O)N(C)Cc1cc(-c2ccc(OC(F)(F)F)cc2)c2c(c1CO)CCO2 | Homo sapiens | CHEMBL5369244 | single protein format | |
CHEMBL5419829 | IC50 | = | 8.0 | nM | 429.42 | C=CS(=O)(=O)NCc1cc(-c2ccc(OC(F)(F)F)cc2)c2c(c1CO)CCO2 | Homo sapiens | CHEMBL5369244 | single protein format | |
CHEMBL5400400 | IC50 | = | 9.0 | nM | 429.4 | Cn1cnc2c(-c3ccc(OC(F)(F)F)cc3)nc(C3CN(C(=O)C4=CCC4)C3)nc21 | Homo sapiens | CHEMBL5369244 | single protein format | |
CHEMBL5432828 | IC50 | = | 9.0 | nM | 418.38 | C=CC(=O)N1CC(c2nn(-c3ccc(OC(F)(F)F)cc3)c3nccc(CO)c23)C1 | Homo sapiens | CHEMBL5374058 | single protein format | |
CHEMBL5403826 | IC50 | = | 10.0 | nM | 390.32 | C#CC(=O)NCc1nn(-c2ccc(OC(F)(F)F)cc2)c2nccc(CO)c12 | Homo sapiens | CHEMBL5374058 | single protein format | |
CHEMBL5428867 | IC50 | = | 13.0 | nM | 452.82 | O=C(/C=C/CO)N1CC(c2nn(-c3ccc(OC(F)(F)F)cc3)c3nccc(Cl)c23)C1 | Homo sapiens | CHEMBL5374058 | single protein format | |
CHEMBL5416415 | IC50 | = | 93.0 | nM | 429.4 | C=CC(=O)NCc1cc(-c2ccc(OC(F)(F)F)cc2)c2ncn(C)c2c1C#CCO | Homo sapiens | CHEMBL5369244 | single protein format | |
CHEMBL5438096 | IC50 | < | 100.0 | nM | 355.36 | C=CC(=O)Nc1cc(/C=C/[C@H]2CC[C@H](C(F)(F)F)CC2)c(OC)nn1 | Homo sapiens | CHEMBL5360850 | single protein format | |
CHEMBL5409535 | IC50 | < | 100.0 | nM | 317.34 | C=CC(=O)Nc1cc(/C=C/C2CCC(F)(F)CC2)c(C#N)cn1 | Homo sapiens | CHEMBL5360850 | single protein format | |
CHEMBL5430925 | IC50 | < | 100.0 | nM | 351.37 | C=CC(=O)Nc1cc(/C=C/C2CCC(F)(F)CC2)c2c(c1F)CCO2 | Homo sapiens | CHEMBL5360850 | single protein format | |
CHEMBL5421419 | IC50 | = | 160.0 | nM | 288.39 | C=CC(=O)N1CCCN(CCCOCc2ccccc2)C1 | Homo sapiens | CHEMBL5360855 | cell-based format | |
CHEMBL5428462 | IC50 | = | 610.0 | nM | 259.35 | C=CC(=O)N1CCC(CCOc2ccccc2)CC1 | Homo sapiens | CHEMBL5360855 | cell-based format |