Q96T60 | PNKP_HUMAN | Bifunctional polynucleotide phosphatase/kinase (PNKP)

Helixβ‑strandTurn secondary structure

Pfam Domain Table

AccessionDomainRangeColor
PF08645PNK3P166–328
PF13671AAA_33367–489
PF17913FHA_211–80

 3D structures mapped by conservation among orthologs

[ Domain: "SMAD/FHA domain" // FHA_1 ]

 PyMOL session


 [ Alpha Fold Model ] (go)



 Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL4303462 IC50 = 60.0 nM 534.66 CCCCCCCCCCC(O)C1C=CC2C(=O)N(c3ccccc3)C(=O)C2N1Nc1ccc([N+](=O)[O-])cc1 Homo sapiens CHEMBL4419662 single protein format
CHEMBL4450001 IC50 = 300.0 nM 560.56 COc1cc(C(O)C2C=CC3C(=O)N(c4ccccc4)C(=O)C3N2Nc2ccc([N+](=O)[O-])cc2)cc(OC)c1OC Homo sapiens CHEMBL4419662 single protein format