Q96PN8 | TSSK3_HUMAN | Testis-specific serine/threonine-protein kinase 3 (TSSK3)

Pfam Domain Table

AccessionDomainRangeColor
PF00069Pkinase - Protein kinase domain10~265

3D structures mapped by conservation among orthologs


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL388978 IC50 = 7.01 nM 466.54 CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 Homo sapiens CHEMBL4328641 single protein format
CHEMBL2334586 IC50 = 91.0 nM 332.41 CC(C)(O)C#Cc1ccc2[nH]c3c(c2c1)-c1nc(N)ncc1CCC3 Homo sapiens CHEMBL5111452 assay format
CHEMBL3943181 IC50 = 420.0 nM 351.41 NC(=O)c1ncc(N[C@@H]2CCCC[C@@H]2N)nc1-c1nc2ccccc2[nH]1 Homo sapiens CHEMBL3865681 single protein format
CHEMBL3415608 IC50 = 420.0 nM 350.43 NC(=O)c1ncc(N[C@@H]2CCCC[C@@H]2N)cc1-c1nc2ccccc2[nH]1 Homo sapiens CHEMBL3418524 single protein format