Q96K76 | UBP47_HUMAN | Ubiquitin carboxyl-terminal hydrolase 47 (USP47)

Helixβ‑strandTurn secondary structure

Pfam Domain Table

AccessionDomainRangeColor
PF00443UCH188–561
PF19718USP47_C1124–1363

 3D structures mapped by conservation among orthologs


 [ Alpha Fold Model ] (go)



 Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL2159507 IC50 = 350.0 nM 507.47 CN(C)CCCOc1ccc(NC(=O)c2cc(C#N)c(Sc3c(Cl)cncc3Cl)s2)cc1 Homo sapiens CHEMBL2162865 single protein format
CHEMBL2398212 IC50 = 400.0 nM 266.65 N#Cc1nc2c(nc1C#N)-c1ccc(Cl)cc1C2=O Homo sapiens CHEMBL5234065 single protein format
CHEMBL2159505 IC50 = 500.0 nM 504.4 CS(=O)(=O)c1ccc(NC(=O)c2cc([N+](=O)[O-])c(Sc3c(Cl)cncc3Cl)s2)cc1 Homo sapiens CHEMBL2162865 single protein format
CHEMBL2159503 IC50 = 530.0 nM 527.46 CN(C)CCCOc1ccc(NC(=O)c2cc([N+](=O)[O-])c(Sc3c(Cl)cncc3Cl)s2)cc1 Homo sapiens CHEMBL2162865 single protein format
CHEMBL2159504 IC50 = 870.0 nM 456.33 COc1ccc(NC(=O)c2cc([N+](=O)[O-])c(Sc3c(Cl)cncc3Cl)s2)cc1 Homo sapiens CHEMBL2162865 single protein format
CHEMBL2159508 IC50 = 1000.0 nM 484.41 CS(=O)(=O)c1ccc(NC(=O)c2cc(C#N)c(Sc3c(Cl)cncc3Cl)s2)cc1 Homo sapiens CHEMBL2162865 single protein format