Q96BR1 | SGK3_HUMAN | Serine/threonine-protein kinase Sgk3 (SGK3)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00069 | Pkinase - Protein kinase domain | 164~419 | |
PF00433 | Pkinase_C - Protein kinase C terminal domain | 440~487 | |
PF00787 | PX - PX domain | 42~119 |
3D structures mapped by conservation among orthologs
[ Domain: "PX domain" // PX ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL3544960 | IC50 | = | 50.0 | nM | 313.79 | NC[C@@](O)(c1ccc(Cl)cc1)c1ccc(-c2cn[nH]c2)cc1 | Homo sapiens | CHEMBL5257196 | single protein format | |
CHEMBL388978 | IC50 | = | 76.5 | nM | 466.54 | CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 | Homo sapiens | CHEMBL4328602 | single protein format | |
CHEMBL5082336 | IC50 | = | 211.0 | nM | 425.86 | N#Cc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(-c2ncc3c(N)n[nH]c3n2)cc1 | Homo sapiens | CHEMBL5043749 | single protein format |