Q96BR1 | SGK3_HUMAN | Serine/threonine-protein kinase Sgk3 (SGK3)

Pfam Domain Table

AccessionDomainRangeColor
PF00069Pkinase - Protein kinase domain164~419
PF00433Pkinase_C - Protein kinase C terminal domain440~487
PF00787PX - PX domain42~119

3D structures mapped by conservation among orthologs

[ Domain: "PX domain" // PX ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL3544960 IC50 = 50.0 nM 313.79 NC[C@@](O)(c1ccc(Cl)cc1)c1ccc(-c2cn[nH]c2)cc1 Homo sapiens CHEMBL5257196 single protein format
CHEMBL388978 IC50 = 76.5 nM 466.54 CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 Homo sapiens CHEMBL4328602 single protein format
CHEMBL5082336 IC50 = 211.0 nM 425.86 N#Cc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(-c2ncc3c(N)n[nH]c3n2)cc1 Homo sapiens CHEMBL5043749 single protein format