Q969H4 | CNKR1_HUMAN | Connector enhancer of kinase suppressor of ras 1 (CNKSR1)

Pfam Domain Table

AccessionDomainRangeColor
PF00169PH - PH domain406~501
PF10534CRIC_ras_sig - Connector enhancer of kinase suppressor of ras78~160

3D structures mapped by conservation among orthologs

[ Domain: "SAM domain-like" // SAM_1_1 ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL4285086 IC50 = 1000.0 nM 369.42 COc1c(/C=C/CO)c(NS(=O)(=O)c2cccs2)cc2c1OCO2 Homo sapiens CHEMBL4257055 assay format
CHEMBL4288751 IC50 = 1000.0 nM 411.46 CCOC(=O)/C=C/c1c(NS(=O)(=O)c2cccs2)cc2c(c1OC)OCO2 Homo sapiens CHEMBL4257055 assay format