Q93096 | TP4A1_HUMAN | Protein tyrosine phosphatase type IVA 1 (PTP4A1)

Pfam Domain Table

AccessionDomainRangeColor
PF22785Tc-R-P - Polymorphic toxin system, DSP-PTPase phosphatase28~123

3D structures mapped by conservation among orthologs

[ Domain: "(Phosphotyrosine protein) phosphatases II" // DSPc ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL4445621 IC50 = 50.0 nM 256.29 N=C1C(=O)NC(=O)c2cc(-c3ccccc3)sc21 Homo sapiens CHEMBL4434554 assay format
CHEMBL3393171 IC50 = 173.0 nM 242.3 Nc1c[nH]c(=O)c2cc(-c3ccccc3)sc12 Homo sapiens CHEMBL3395567 assay format
CHEMBL55 IC50 = 300.0 nM 340.43 N=C(N)c1ccc(OCCCCCOc2ccc(C(=N)N)cc2)cc1 Homo sapiens CHEMBL4434545 single protein format
CHEMBL1088572 IC50 = 676.0 nM 387.24 O=P([O-])(O)OC1C=C(c2ccccc2F)Nc2cc3c(cc21)OCO3.[Na+] Homo sapiens CHEMBL1113392 single protein format