Q92570 | NR4A3_HUMAN | Nuclear receptor subfamily 4 group A member 3 (NR4A3)

Pfam Domain Table

AccessionDomainRangeColor
PF00104Hormone_recep - Ligand-binding domain of nuclear hormone receptor434~606
PF00105zf-C4 - Double treble clef zinc finger, C4 type291~359

3D structures mapped by conservation among orthologs


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL4560385 IC50 = 1.2 nM 438.44 N#CN1CCC[C@@H](n2nc(-c3ccc(Oc4ccc(F)cc4F)cc3)c(C(N)=O)c2N)C1 Homo sapiens CHEMBL5243497 single protein format
CHEMBL5404368 IC50 = 18.0 nM 465.52 C=CC(=O)N1CC[C@@H](N2N=C(Nc3ccc(Oc4ccccc4)cc3)c3c[nH]c4ncnc2c34)C1 Homo sapiens CHEMBL5355222 single protein format
CHEMBL1873475 IC50 = 78.0 nM 440.51 C=CC(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1 Homo sapiens CHEMBL4720218 single protein format
CHEMBL4755698 IC50 = 210.6 nM 405.46 C=CC(=O)N1CCC(Cn2cc(-c3ccc4c(c3)OCO4)c3c(N)ncnc32)CC1 Homo sapiens CHEMBL4720218 single protein format