Q8WYB5 | KAT6B_HUMAN | Histone acetyltransferase KAT6B (KAT6B)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00628 | PHD - PHD-finger | 272~317 | |
PF01853 | MOZ_SAS - MOZ/SAS family | 776~952 | |
PF17772 | zf-MYST - MYST family zinc finger domain | 718~771 | |
PF21524 | SAMD1_WH - SAM domain-containing protein 1, WH domain | 11~73 |
3D structures mapped by conservation among orthologs
[ Domain: "FYVE/PHD zinc finger" // PHD ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL4456585 | IC50 | = | 6.3 | nM | 389.38 | O=C(NNS(=O)(=O)c1ccccc1F)c1cc(F)cc(-c2ccccn2)c1 | Homo sapiens | CHEMBL5210226 | single protein format | |
CHEMBL4455897 | IC50 | = | 28.0 | nM | 384.43 | Cc1cc(-c2ccccc2)cc(C(=O)NNS(=O)(=O)c2ccccc2)c1F | Homo sapiens | CHEMBL4374940 | cell-based format |