Q8WYB5 | KAT6B_HUMAN | Histone acetyltransferase KAT6B (KAT6B)

Helixβ‑strandTurn secondary structure

Pfam Domain Table

AccessionDomainRangeColor
PF00628PHD272–317
PF01853MOZ_SAS776–952
PF17772zf-MYST718–771
PF21524SAMD1_WH11–73

 3D structures mapped by conservation among orthologs

[ Domain: "FYVE/PHD zinc finger" // PHD ]

 PyMOL session


 [ Alpha Fold Model ] (go)



 Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL4456585 IC50 = 6.3 nM 389.38 O=C(NNS(=O)(=O)c1ccccc1F)c1cc(F)cc(-c2ccccn2)c1 Homo sapiens CHEMBL5210226 single protein format
CHEMBL4455897 IC50 = 28.0 nM 384.43 Cc1cc(-c2ccccc2)cc(C(=O)NNS(=O)(=O)c2ccccc2)c1F Homo sapiens CHEMBL4374940 cell-based format