Q6DT37 | MRCKG_HUMAN | Serine/threonine-protein kinase MRCK gamma (CDC42BPG)

Helixβ‑strandTurn secondary structure

Pfam Domain Table

AccessionDomainRangeColor
PF00069Pkinase71–337
PF00130C1_1879–927
PF00433Pkinase_C357–398
PF00780CNH1103–1360
PF08826DMPK_coil744–800
PF25346PH_MRCK942–1066

 3D structures mapped by conservation among orthologs


 [ Alpha Fold Model ] (go)



 Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL388978 IC50 = 0.848 nM 466.54 CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 Homo sapiens CHEMBL4328388 single protein format