Q6DT37 | MRCKG_HUMAN | Serine/threonine-protein kinase MRCK gamma (CDC42BPG)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00069 | Pkinase - Protein kinase domain | 71~337 | |
PF00130 | C1_1 - Phorbol esters/diacylglycerol binding domain (C1 domain) | 879~927 | |
PF00433 | Pkinase_C - Protein kinase C terminal domain | 357~398 | |
PF00780 | CNH - CNH domain | 1103~1360 | |
PF08826 | DMPK_coil - DMPK coiled coil domain like | 744~800 | |
PF25346 | PH_MRCK - MRCK kinase PH domain | 942~1066 |
3D structures mapped by conservation among orthologs
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL388978 | IC50 | = | 0.848 | nM | 466.54 | CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 | Homo sapiens | CHEMBL4328388 | single protein format |