Q6DT37 | MRCKG_HUMAN | Serine/threonine-protein kinase MRCK gamma (CDC42BPG)

Pfam Domain Table

AccessionDomainRangeColor
PF00069Pkinase - Protein kinase domain71~337
PF00130C1_1 - Phorbol esters/diacylglycerol binding domain (C1 domain)879~927
PF00433Pkinase_C - Protein kinase C terminal domain357~398
PF00780CNH - CNH domain1103~1360
PF08826DMPK_coil - DMPK coiled coil domain like744~800
PF25346PH_MRCK - MRCK kinase PH domain942~1066

3D structures mapped by conservation among orthologs


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL388978 IC50 = 0.848 nM 466.54 CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 Homo sapiens CHEMBL4328388 single protein format