Q16621 | NFE2_HUMAN | Transcription factor NF-E2 45 kDa subunit (NFE2)

Pfam Domain Table

AccessionDomainRangeColor
PF03131bZIP_Maf - bZIP Maf transcription factor239~329

3D structures mapped by conservation among orthologs

[ Domain: "A DNA-binding domain in eukaryotic transcription factors" // bZIP_Maf ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL4555143 IC50 = 71.2 nM 433.54 CC(C)(C)c1cc(NC(=O)CSc2nnnn2-c2ccccc2)n(-c2ccccc2)n1 Homo sapiens CHEMBL4400009 assay format
CHEMBL4447685 IC50 = 112.6 nM 445.48 CC(C)(C)c1cc(NC(=O)COC(=O)c2ccc(-n3cnnn3)cc2)n(-c2ccccc2)n1 Homo sapiens CHEMBL4400009 assay format