Q16620 | NTRK2_HUMAN | BDNF/NT-3 growth factors receptor (NTRK2)

Helixβ‑strandTurn secondary structure

Pfam Domain Table

AccessionDomainRangeColor
PF01462LRRNT31–60
PF07679I-set204–283
PF07679I-set306–374
PF07714PK_Tyr_Ser-Thr539–806
PF13855LRR_892–149
PF16920LRRCT_2151–195

 3D structures mapped by conservation among orthologs

[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // I-set_11 ]

 PyMOL session

[ Domain: "Protein kinase" // Pkinase_Tyr ]

 PyMOL session


 [ Alpha Fold Model ] (go)



 Known binders annotated in ChEMBL

 Ki CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL3286829 Ki = 0.4 nM 421.48 C[C@H]1Oc2cc(cnc2N)-c2c(C3CC3)nn(C)c2CN(C)C(=O)c2ccc(F)cc21 Homo sapiens CHEMBL3293393 single protein format
CHEMBL3286820 Ki = 0.5 nM 395.44 Cc1nn(C)c2c1-c1cnc(N)c(c1)O[C@H](C)c1cc(F)ccc1C(=O)N(C)C2 Homo sapiens CHEMBL3293393 single protein format
CHEMBL5088153 Ki = 1.0 nM 575.07 Cc1cc(NC(=O)Nc2cc(C(C)(C)C)nn2-c2ccc(Cl)cc2)ccc1Nc1ncnc2c1OC(C)(C)C(=O)N2 Homo sapiens CHEMBL5045136 single protein format
CHEMBL3286830 Ki = 23.0 nM 406.42 C[C@H]1Oc2cc(cnc2N)-c2c(nn(C)c2C#N)CN(C)C(=O)c2ccc(F)cc21 Homo sapiens CHEMBL3293393 single protein format
CHEMBL3286832 Ki = 65.0 nM 443.44 C[C@H]1Oc2nc(cnc2N)-c2c(nc3ccc(C#N)cn23)CN(C)C(=O)c2ccc(F)cc21 Homo sapiens CHEMBL3293393 single protein format
CHEMBL3286831 Ki = 77.0 nM 432.46 Cc1cnc2nc3c(n2c1)-c1cnc(N)c(c1)O[C@H](C)c1cc(F)ccc1C(=O)N(C)C3 Homo sapiens CHEMBL3293393 single protein format