Q15717 | ELAV1_HUMAN | ELAV-like protein 1 (ELAVL1)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00076 | RRM_1 - RNA recognition motif | 22~92 | |
PF00076 | RRM_1 - RNA recognition motif | 108~174 | |
PF00076 | RRM_1 - RNA recognition motif | 246~314 |
3D structures mapped by conservation among orthologs
[ Domain: "RNA-binding domain, RBD" // RRM_1 ]
[ Domain: "RNA-binding domain, RBD" // RRM_1_2 ]
[ Domain: "RNA-binding domain, RBD" // RRM_1_4 ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL227075 | IC50 | = | 68.0 | nM | 278.31 | Cc1cccc2c3c(ccc12)C1=C(C(=O)C3=O)[C@@H](C)CO1 | Homo sapiens | CHEMBL4018390 | single protein format | |
CHEMBL4061748 | IC50 | = | 380.0 | nM | 508.56 | N#Cc1c(N)nc(SCC(=O)c2ccc(O)c(O)c2)c(C#N)c1-c1ccc(COc2ccccc2)cc1 | Homo sapiens | CHEMBL4018388 | single protein format | |
CHEMBL4075458 | Ki | = | 12.8 | nM | 363.39 | O=C1C=Cc2c(c(-c3ccccc3)cn2S(=O)(=O)c2ccccc2)C1=O | Homo sapiens | CHEMBL4059046 | assay format | |
CHEMBL4064932 | Ki | = | 15.0 | nM | 501.59 | COc1ccc(SC2=CC(=O)C(=O)c3c(-c4ccccc4)cn(S(=O)(=O)c4ccccc4)c32)cc1 | Homo sapiens | CHEMBL4059046 | assay format | |
CHEMBL4095060 | Ki | = | 41.0 | nM | 469.52 | COc1ccc(C2=CC(=O)C(=O)c3c(-c4ccccc4)cn(S(=O)(=O)c4ccccc4)c32)cc1 | Homo sapiens | CHEMBL4059046 | assay format | |
CHEMBL4100171 | Ki | = | 48.0 | nM | 381.38 | O=C1C=Cc2c(c(-c3ccccc3)cn2S(=O)(=O)c2ccc(F)cc2)C1=O | Homo sapiens | CHEMBL4059046 | assay format | |
CHEMBL227075 | Ki | = | 50.0 | nM | 278.31 | Cc1cccc2c3c(ccc12)C1=C(C(=O)C3=O)[C@@H](C)CO1 | Homo sapiens | CHEMBL4059046 | assay format | |
CHEMBL4105230 | Ki | = | 55.0 | nM | 469.52 | COc1cccc(C2=CC(=O)C(=O)c3c(-c4ccccc4)cn(S(=O)(=O)c4ccccc4)c32)c1 | Homo sapiens | CHEMBL4059046 | assay format | |
CHEMBL4073526 | Ki | = | 56.0 | nM | 301.32 | CS(=O)(=O)n1cc(-c2ccccc2)c2c1C=CC(=O)C2=O | Homo sapiens | CHEMBL4059046 | assay format | |
CHEMBL4094161 | Ki | = | 81.0 | nM | 420.45 | CC(=O)Nc1ccc(S(=O)(=O)n2cc(-c3ccccc3)c3c2C=CC(=O)C3=O)cc1 | Homo sapiens | CHEMBL4059046 | assay format | |
CHEMBL1499653 | Ki | = | 350.0 | nM | 513.59 | COc1ccc(C(CC(=O)N2CCCC2)c2c(OC)cc(OC)c3c(-c4ccccc4)cc(=O)oc23)cc1 | Homo sapiens | CHEMBL4018391 | single protein format | |
CHEMBL1522581 | Ki | = | 570.0 | nM | 515.61 | CCN(CC)C(=O)CC(c1ccc(OC)cc1)c1c(OC)cc(OC)c2c(-c3ccccc3)cc(=O)oc12 | Homo sapiens | CHEMBL4018391 | single protein format | |
CHEMBL1330249 | Ki | = | 590.0 | nM | 575.66 | CCN(CC)C(=O)CC(c1cc(OC)c(OC)c(OC)c1)c1c(OC)cc(OC)c2c(-c3ccccc3)cc(=O)oc12 | Homo sapiens | CHEMBL4018391 | single protein format | |
CHEMBL1390568 | Ki | = | 800.0 | nM | 529.59 | COc1ccc(C(CC(=O)N2CCOCC2)c2c(OC)cc(OC)c3c(-c4ccccc4)cc(=O)oc23)cc1 | Homo sapiens | CHEMBL4018391 | single protein format |