Q15078 | CD5R1_HUMAN | Cyclin-dependent kinase 5 activator 1 (CDK5R1)
Pfam Domain Table
| Accession | Domain | Range | Color |
|---|---|---|---|
| PF03261 | CDK5_activator - Cyclin-dependent kinase 5 activator protein | 136~293 |
3D structures mapped by conservation among orthologs
[ Domain: "Cyclin-like" // CDK5_activator ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
| molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
|---|---|---|---|---|---|---|---|---|---|---|
| CHEMBL440411 |  |
IC50 | = | 7.0 | nM | 357.35 | O=C1Nc2ccc(S(=O)(=O)O)cc2/C1=C1/Nc2ccccc2/C1=N\O | Homo sapiens | CHEMBL937655 | single protein format |
| CHEMBL337300 |  |
IC50 | = | 20.0 | nM | 403.18 | O=Nc1c(-c2c(O)[nH]c3ccc(I)cc23)[nH]c2ccccc12 | Homo sapiens | CHEMBL937655 | single protein format |
| CHEMBL126077 |  |
IC50 | = | 100.0 | nM | 277.28 | O=Nc1c(-c2c(O)[nH]c3ccccc23)[nH]c2ccccc12 | Homo sapiens | CHEMBL937655 | single protein format |