Q13555 | KCC2G_HUMAN | Calcium/calmodulin-dependent protein kinase type II subunit gamma (CAMK2G)

Pfam Domain Table

AccessionDomainRangeColor
PF00069Pkinase - Protein kinase domain14~272
PF08332CaMKII_AD - Calcium/calmodulin dependent protein kinase II association domain426~553

3D structures mapped by conservation among orthologs

[ Domain: "NTF2-like" // DUF4440 ]

 PyMOL session

[ Domain: "Protein kinase" // Pkinase_Tyr ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL388978 IC50 = 0.387 nM 466.54 CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 Homo sapiens CHEMBL4328336 single protein format
CHEMBL3975634 IC50 = 0.7 nM 452.51 CN[C@H]1CC2OC([C@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(O)=NC4 Homo sapiens CHEMBL3707764 single protein format
CHEMBL288441 IC50 = 184.0 nM 530.46 COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(C)CC4)c(OC)cc23)c(Cl)cc1Cl Homo sapiens CHEMBL1244345 single protein format
CHEMBL4556306 IC50 = 790.0 nM 429.58 COc1ccc(S(=O)(=O)N(CCCC(=O)C2CCCCCC2)c2ccccc2)cc1 Homo sapiens CHEMBL5131908 single protein format
CHEMBL5303487 IC50 = 1000.0 nM 398.89 COc1cc(-c2cn[nH]c2)ccc1C(=O)Nc1ccc2c(c1)CCNCC2.Cl Homo sapiens CHEMBL5478972 single protein format