Q13555 | KCC2G_HUMAN | Calcium/calmodulin-dependent protein kinase type II subunit gamma (CAMK2G)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00069 | Pkinase - Protein kinase domain | 14~272 | |
PF08332 | CaMKII_AD - Calcium/calmodulin dependent protein kinase II association domain | 426~553 |
3D structures mapped by conservation among orthologs
[ Domain: "NTF2-like" // DUF4440 ]
[ Domain: "Protein kinase" // Pkinase_Tyr ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL388978 | IC50 | = | 0.387 | nM | 466.54 | CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 | Homo sapiens | CHEMBL4328336 | single protein format | |
CHEMBL3975634 | IC50 | = | 0.7 | nM | 452.51 | CN[C@H]1CC2OC([C@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(O)=NC4 | Homo sapiens | CHEMBL3707764 | single protein format | |
CHEMBL288441 | IC50 | = | 184.0 | nM | 530.46 | COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(C)CC4)c(OC)cc23)c(Cl)cc1Cl | Homo sapiens | CHEMBL1244345 | single protein format | |
CHEMBL4556306 | IC50 | = | 790.0 | nM | 429.58 | COc1ccc(S(=O)(=O)N(CCCC(=O)C2CCCCCC2)c2ccccc2)cc1 | Homo sapiens | CHEMBL5131908 | single protein format | |
CHEMBL5303487 | IC50 | = | 1000.0 | nM | 398.89 | COc1cc(-c2cn[nH]c2)ccc1C(=O)Nc1ccc2c(c1)CCNCC2.Cl | Homo sapiens | CHEMBL5478972 | single protein format |