Q13554 | KCC2B_HUMAN | Calcium/calmodulin-dependent protein kinase type II subunit beta (CAMK2B)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00069 | Pkinase - Protein kinase domain | 14~272 | |
PF08332 | CaMKII_AD - Calcium/calmodulin dependent protein kinase II association domain | 534~661 |
3D structures mapped by conservation among orthologs
[ Domain: "Protein kinase" // Pkinase_Tyr ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL388978 | IC50 | = | 0.07 | nM | 466.54 | CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 | Homo sapiens | CHEMBL4145856 | single protein format | |
CHEMBL1231206 | IC50 | = | 70.0 | nM | 374.47 | Cc1ccc(-c2ccc3c(ccc4sc5c(c43)NC[C@@H](C)NC5=O)n2)cn1 | Homo sapiens | CHEMBL5212744 | single protein format | |
CHEMBL1945559 | IC50 | = | 83.0 | nM | 363.25 | Cn1c2c(c3ccc(Cl)c(Cl)c31)C(C#N)C1(CCNCC1)NC2=O | Homo sapiens | CHEMBL1947302 | single protein format |