Q03431 | PTH1R_HUMAN | Parathyroid hormone/parathyroid hormone-related peptide receptor (PTH1R)

Pfam Domain Table

AccessionDomainRangeColor
PF000027tm_2 - 7 transmembrane receptor (Secretin family)186~455
PF02793HRM - Hormone receptor domain107~172

3D structures mapped by conservation among orthologs

[ Domain: "Family A G protein-coupled receptor-like" // 7tm_2 ]

 PyMOL session

[ Domain: "UDP-Glycosyltransferase/glycogen phosphorylase" // Glycos_transf_1 ]

 PyMOL session

[ Domain: "Hormone receptor domain (HRM, Pfam 02793)" // HRM ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL515170 IC50 = 990.0 nM 361.31 CC[C@@H]1O[C@](/C=C/C2CC2)(C(F)(F)F)c2c(ccc(F)c2F)NC1=O Homo sapiens CHEMBL944465 cell-based format