Q03431 | PTH1R_HUMAN | Parathyroid hormone/parathyroid hormone-related peptide receptor (PTH1R)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00002 | 7tm_2 - 7 transmembrane receptor (Secretin family) | 186~455 | |
PF02793 | HRM - Hormone receptor domain | 107~172 |
3D structures mapped by conservation among orthologs
[ Domain: "Family A G protein-coupled receptor-like" // 7tm_2 ]
[ Domain: "UDP-Glycosyltransferase/glycogen phosphorylase" // Glycos_transf_1 ]
[ Domain: "Hormone receptor domain (HRM, Pfam 02793)" // HRM ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL515170 | IC50 | = | 990.0 | nM | 361.31 | CC[C@@H]1O[C@](/C=C/C2CC2)(C(F)(F)F)c2c(ccc(F)c2F)NC1=O | Homo sapiens | CHEMBL944465 | cell-based format |