Q00532 | CDKL1_HUMAN | Cyclin-dependent kinase-like 1 (CDKL1)

Pfam Domain Table

AccessionDomainRangeColor
PF00069Pkinase - Protein kinase domain4~287

3D structures mapped by conservation among orthologs

[ Domain: "Protein kinase" // Pkinase_Tyr ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL455428 IC50 = 60.0 nM 368.42 CNC(=O)c1ccc(Nc2nccc(-c3cnc(C)n3C(C)C)n2)cc1F Homo sapiens CHEMBL1022595 single protein format