P54762 | EPHB1_HUMAN | Ephrin type-B receptor 1 (EPHB1)
Pfam Domain Table
Accession | Domain | Range | Color |
---|---|---|---|
PF00041 | fn3 - Fibronectin type III domain | 326~415 | |
PF00041 | fn3 - Fibronectin type III domain | 443~519 | |
PF00536 | SAM_1 - SAM domain (Sterile alpha motif) | 911~973 | |
PF01404 | Ephrin_lbd - Ephrin receptor ligand binding domain | 20~196 | |
PF07714 | PK_Tyr_Ser-Thr - Protein tyrosine and serine/threonine kinase | 619~878 | |
PF14575 | EphA2_TM - Ephrin type-A receptor 2 transmembrane domain | 542~616 | |
PF25599 | Ephrin_CRD - Ephrin cysteine rich domain | 197~255 |
3D structures mapped by conservation among orthologs
[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // fn3 ]
[ Domain: "SAM domain-like" // SAM_1 ]
[ Domain: "Protein kinase" // Pkinase_Tyr ]
[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
Only the first 20 rows are shown.
molecule_chembl_id | structure | assay_type | relation | value | unit | mol_wt | smiles | organism | assay_chembl_id | bao_label |
---|---|---|---|---|---|---|---|---|---|---|
CHEMBL566515 | IC50 | = | 1.1 | nM | 417.43 | COc1ccccc1-n1c(-c2cc(O)ccc2C)cn2c3c(=O)[nH]c(=O)n(C)c3nc12 | Homo sapiens | CHEMBL1046777 | single protein format | |
CHEMBL488840 | IC50 | = | 6.0 | nM | 417.45 | Cc1cccc(C)c1/C=C/n1cnc2c(Nc3ccc(P(C)(C)=O)cc3)ncnc21 | Homo sapiens | CHEMBL976279 | single protein format | |
CHEMBL4846921 | IC50 | = | 29.8 | nM | 508.67 | CCN1CCN(c2ccc(Nc3ncc4scc(-c5cccc(NS(C)(=O)=O)c5)c4n3)cc2)CC1 | Homo sapiens | CHEMBL4839037 | single protein format | |
CHEMBL103667 | IC50 | = | 110.0 | nM | 527.67 | Cc1ccc(-n2nc(C(C)(C)C)cc2NC(=O)Nc2ccc(OCCN3CCOCC3)c3ccccc23)cc1 | Homo sapiens | CHEMBL1932847 | single protein format | |
CHEMBL388978 | IC50 | = | 127.9 | nM | 466.54 | CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 | Homo sapiens | CHEMBL3820483 | single protein format | |
CHEMBL4793380 | IC50 | = | 388.0 | nM | 423.48 | CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4c3OCCCN4)cc2)no1 | Homo sapiens | CHEMBL4767004 | single protein format | |
CHEMBL5425418 | IC50 | = | 632.0 | nM | 359.38 | CNc1ncc2cc(-c3cc(F)ccc3F)c(=O)n(CCCCN)c2n1 | Homo sapiens | CHEMBL5327128 | cell-based format |