P42679 | MATK_HUMAN | Megakaryocyte-associated tyrosine-protein kinase (MATK)

Pfam Domain Table

AccessionDomainRangeColor
PF00017SH2 - SH2 domain122~196
PF00018SH3_1 - SH3 domain64~99
PF07714PK_Tyr_Ser-Thr - Protein tyrosine and serine/threonine kinase236~478

3D structures mapped by conservation among orthologs

[ Domain: "SH3" // SH3_1 ]

 PyMOL session

[ Domain: "SH2" // SH2 ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL388978 IC50 = 492.0 nM 466.54 CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 Homo sapiens CHEMBL4328379 single protein format