P24046 | GBRR1_HUMAN | Gamma-aminobutyric acid receptor subunit rho-1 (GABRR1)

Pfam Domain Table

AccessionDomainRangeColor
PF02931Neur_chan_LBD - Neurotransmitter-gated ion-channel ligand binding domain81~280
PF02932Neur_chan_memb - Neurotransmitter-gated ion-channel transmembrane region288~475

3D structures mapped by conservation among orthologs


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL15891 IC50 = 91.0 nM 290.83 Cl[C@H]1[C@H](Cl)[C@@H](Cl)[C@@H](Cl)[C@H](Cl)[C@H]1Cl Homo sapiens CHEMBL3073008 single protein format
CHEMBL1890408 IC50 = 800.0 nM 406.93 O=S1OC[C@@H]2[C@H](CO1)[C@@]1(Cl)C(Cl)=C(Cl)[C@]2(Cl)C1(Cl)Cl Homo sapiens CHEMBL3073008 single protein format