P23470 | PTPRG_HUMAN | Receptor-type tyrosine-protein phosphatase gamma (PTPRG)

Pfam Domain Table

AccessionDomainRangeColor
PF00041fn3 - Fibronectin type III domain348~429
PF00102Y_phosphatase - Protein-tyrosine phosphatase874~1118
PF00102Y_phosphatase - Protein-tyrosine phosphatase1175~1408
PF00194Carb_anhydrase - Eukaryotic-type carbonic anhydrase67~320

3D structures mapped by conservation among orthologs

[ Domain: "Carbonic anhydrase" // Carb_anhydrase ]

 PyMOL session

[ Domain: "(Phosphotyrosine protein) phosphatases II" // Y_phosphatase ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL1910889 IC50 = 500.0 nM 532.45 COc1ccc(S(=O)(=O)NC(=O)c2sccc2SCc2ccc(Cl)c(Cl)c2)cc1C(=O)O Homo sapiens CHEMBL1914005 assay format