P14616 | INSRR_HUMAN | Insulin receptor-related protein (INSRR)

Helixβ‑strandTurn secondary structure

Pfam Domain Table

AccessionDomainRangeColor
PF00041fn3820–905
PF00757Furin-like174–329
PF01030Recep_L_domain47–157
PF01030Recep_L_domain346–454
PF07714PK_Tyr_Ser-Thr980–1245

 3D structures mapped by conservation among orthologs


 [ Alpha Fold Model ] (go)



 Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL388978 IC50 = 15.0 nM 466.54 CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 Homo sapiens CHEMBL4328456 single protein format
CHEMBL1091644 IC50 = 75.0 nM 421.5 C[C@]1(O)C[C@@H](c2nc(-c3ccc4ccc(-c5ccccc5)nc4c3)c3c(N)nccn32)C1 Homo sapiens CHEMBL5210320 single protein format