P11274 | BCR_HUMAN | Breakpoint cluster region protein (BCR)

Helixβ‑strandTurn secondary structure

Pfam Domain Table

AccessionDomainRangeColor
PF00168C2913–1007
PF00620RhoGAP1068–1215
PF00621RhoGEF503–689
PF09036Bcr-Abl_Oligo3–75
PF19057PH_19703–781

 3D structures mapped by conservation among orthologs

[ Domain: "PH domain-like" // PH_10 ]

 PyMOL session

[ Domain: "DBL homology domain (DH-domain)" // RhoGEF ]

 PyMOL session

[ Domain: "Bcr-Abl oncoprotein oligomerization domain" // Bcr-Abl_Oligo ]

 PyMOL session

[ Domain: "Bcr-Abl oncoprotein oligomerization domain" // Bcr-Abl_Oligo ]

 PyMOL session


 [ Alpha Fold Model ] (go)



 Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL434335 IC50 = 573.0 nM 439.52 Cc1ccc(NC(=O)Nc2cccc(N(C)C)c2)cc1Nc1nccc(-c2cccnc2)n1 Homo sapiens CHEMBL832728 single protein format
CHEMBL184742 IC50 = 720.0 nM 465.56 Cc1ccc(NC(=O)Nc2cccc(N3CCCC3)c2)cc1Nc1nccc(-c2cccnc2)n1 Homo sapiens CHEMBL832728 single protein format