P0DMV8 | HS71A_HUMAN | Heat shock 70 kDa protein 1A (HSPA1A)

Pfam Domain Table

AccessionDomainRangeColor
PF00012HSP70 - Hsp70 protein6~611

3D structures mapped by conservation among orthologs

[ Domain: "Heat shock protein 70kD (HSP70), peptide-binding domain" // HSP70_2nd ]

 PyMOL session

[ Domain: "Heat shock protein 70kD (HSP70), C-terminal subdomain" // HSP70_3rd ]

 PyMOL session

[ Domain: "Ribonuclease H-like" // HSP70_1st ]

 PyMOL session

[ Domain: "Ribonuclease H-like" // MreB_Mbl_C ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL502775 IC50 = 332.0 nM 314.25 O=C(O)/C=C/c1c2ccc(=O)c(O)c-2oc2c(O)c(O)ccc12 Homo sapiens CHEMBL1614297 single protein format
CHEMBL1481974 IC50 = 578.0 nM 316.27 O=C(O)CCc1c2ccc(=O)c(O)c-2oc2c(O)c(O)ccc12 Homo sapiens CHEMBL1614297 single protein format
CHEMBL471004 IC50 = 634.0 nM 394.38 CC1C2C=CC1C(c1c3ccc(=O)c(O)c-3oc3c(O)c(O)ccc13)C2C(=O)O Homo sapiens CHEMBL1614297 single protein format
CHEMBL6246 IC50 = 760.0 nM 302.19 O=c1oc2c(O)c(O)cc3c(=O)oc4c(O)c(O)cc1c4c23 Homo sapiens CHEMBL1614054 single protein format