P0DJD9 | PEPA5_HUMAN | Pepsin A-5 (PGA5)

Pfam Domain Table

AccessionDomainRangeColor
PF00026Asp - Eukaryotic aspartyl protease75~387
PF07966A1_Propeptide - A1 Propeptide19~45

3D structures mapped by conservation among orthologs


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL3142364 IC50 = 700.0 nM 485.71 CCCCCCC(O)[C@H](CCC)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(C)C Homo sapiens CHEMBL759819 single protein format
CHEMBL3142349 IC50 = 790.0 nM 527.79 CCCCCCCCC(O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(C)C Homo sapiens CHEMBL759819 single protein format
CHEMBL63831 IC50 = 830.0 nM 499.74 CCCCCCC(O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(C)C Homo sapiens CHEMBL759819 single protein format
CHEMBL3142354 IC50 = 910.0 nM 457.66 CCCCC(O)[C@H](CCC)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(C)C Homo sapiens CHEMBL759819 single protein format