P08047 | SP1_HUMAN | Transcription factor Sp1 (SP1)

Helixβ‑strandTurn secondary structure

Pfam Domain Table

AccessionDomainRangeColor
PF00096zf-C2H2656–680
PF00096zf-C2H2686–708

 3D structures mapped by conservation among orthologs

[ Domain: "beta-beta-alpha zinc fingers" // zf-C2H2_12 ]

 PyMOL session

[ Domain: "beta-beta-alpha zinc fingers" // zf-C2H2_17 ]

 PyMOL session


 [ Alpha Fold Model ] (go)



 Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL2105734 IC50 = 8.0 nM 443.3 COCC[n+]1c2c(n(Cc3cnccn3)c1C)C(=O)c1ccccc1C2=O.[Br-] Homo sapiens CHEMBL5379429 cell-based format