P00395 | COX1_HUMAN | Cytochrome c oxidase subunit 1 (MT-CO1)

Pfam Domain Table

AccessionDomainRangeColor
PF00115COX1 - Cytochrome C and Quinol oxidase polypeptide I14~460

3D structures mapped by conservation among orthologs

[ Domain: "Cytochrome c oxidase subunit I-like" // COX1 ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL1774043 IC50 = 130.0 nM 576.63 COc1ccc(-c2cnc(C(=O)N3CCN(c4cc(C(=O)O)c5ccccc5c4)CC3)nc2-c2ccc(C)cc2F)cc1 Homo sapiens CHEMBL1775456 single protein format
CHEMBL441414 IC50 = 500.0 nM 248.32 C[C@H](C(=O)O)c1ccc(C[C@H]2CCC[C@@H]2O)cc1 Homo sapiens CHEMBL5162740 single protein format