O95259 | KCNH1_HUMAN | Potassium voltage-gated channel subfamily H member 1 (KCNH1)

Pfam Domain Table

AccessionDomainRangeColor
PF00027cNMP_binding - Cyclic nucleotide-binding domain600~682
PF00520Ion_trans - Ion transport protein219~509
PF13426PAS_9 - PAS domain41~135

3D structures mapped by conservation among orthologs

[ Domain: "sensor domains" // PAS ]

 PyMOL session


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 IC50 CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL3261075 IC50 = 490.0 nM 388.41 C[C@@]1(c2cc(NC(=O)c3ccc(C#N)cn3)ccc2F)Cn2cccc2C(N)=N1 Homo sapiens CHEMBL4307470 single protein format