O15440 | MRP5_HUMAN | ATP-binding cassette sub-family C member 5 (ABCC5)

Pfam Domain Table

AccessionDomainRangeColor
PF00005ABC_tran - ABC transporter578~712
PF00005ABC_tran - ABC transporter1210~1358
PF00664ABC_membrane - ABC transporter transmembrane region179~446
PF00664ABC_membrane - ABC transporter transmembrane region860~1141

3D structures mapped by conservation among orthologs


[ Alpha Fold Model ] (go)



Known binders annotated in ChEMBL

 Ki CSV
Only the first 20 rows are shown.
molecule_chembl_idstructureassay_typerelation valueunitmol_wtsmilesorganism assay_chembl_idbao_label
CHEMBL1338248 Ki = 65.3 nM 527.56 CCCc1nn(C)c2c(O)nc(-c3cc(S(=O)(=O)Nc4ccc(O)c(C(=O)O)c4)ccc3OCC)nc12 Homo sapiens CHEMBL2049559 cell-based format
CHEMBL2047880 Ki = 75.3 nM 541.59 CCOc1ccc(S(=O)(=O)Nc2ccc(O)c(C(=O)O)c2)cc1-c1nc2c(C(C)(C)C)nn(C)c2c(=O)[nH]1 Homo sapiens CHEMBL2049559 cell-based format